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Talabostat mesylate

CAS No. 150080-09-4

Talabostat mesylate ( Val-boroPro (mesylate); PT100 (mesylate )

产品货号. M17326 CAS No. 150080-09-4

Talabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein.

纯度: 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥794 有现货
10MG ¥1288 有现货
50MG ¥3216 有现货
100MG 获取报价 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Talabostat mesylate
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Talabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein.
  • 产品描述
    Talabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein. This agent may also stimulate the production of colony stimulating factors, such as granulocyte colony-stimulating factor (G-CSF), resulting in the stimulation of hematopoiesis.
  • 同义词
    Val-boroPro (mesylate); PT100 (mesylate
  • 通路
    Metabolic Enzyme/Protease
  • 靶点
    Phosphatase
  • 受体
    DPP-4
  • 研究领域
    Metabolic Disease
  • 适应症
    ——

化学信息

  • CAS Number
    150080-09-4
  • 分子量
    310.18
  • 分子式
    C10H23BN2O6S
  • 纯度
    98%
  • 溶解度
    DMSO : ≥ 40 mg/mL. 128.96 mM
  • SMILES
    OB([C@H]1N(C(=O)[C@@H](N)C(C)C)CCC1)O.CS(=O)(=O)O
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Cristillo AD, et al. HIV-1 Env vaccine comprised of electroporated DNA and protein co-administered with Talabostat. Biochem Biophys Res Commun. 2008 May 23;370(1):22-6.
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