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Talabostat mesylate
CAS No. 150080-09-4
Talabostat mesylate ( Val-boroPro (mesylate); PT100 (mesylate )
产品货号. M17326 CAS No. 150080-09-4
Talabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein.
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥794 | 有现货 |
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| 10MG | ￥1288 | 有现货 |
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| 50MG | ￥3216 | 有现货 |
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| 100MG | 获取报价 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Talabostat mesylate
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Talabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein.
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产品描述Talabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein. This agent may also stimulate the production of colony stimulating factors, such as granulocyte colony-stimulating factor (G-CSF), resulting in the stimulation of hematopoiesis.
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同义词Val-boroPro (mesylate); PT100 (mesylate
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通路Metabolic Enzyme/Protease
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靶点Phosphatase
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受体DPP-4
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研究领域Metabolic Disease
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适应症——
化学信息
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CAS Number150080-09-4
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分子量310.18
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分子式C10H23BN2O6S
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纯度98%
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溶解度DMSO : ≥ 40 mg/mL. 128.96 mM
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SMILESOB([C@H]1N(C(=O)[C@@H](N)C(C)C)CCC1)O.CS(=O)(=O)O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Cristillo AD, et al. HIV-1 Env vaccine comprised of electroporated DNA and protein co-administered with Talabostat. Biochem Biophys Res Commun. 2008 May 23;370(1):22-6.
产品手册
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